TELMISARTAN-MEDICINES ABOUT,CHEMICAL FORMULA,USES,MECHANISM,RECOMMENDED DOSAGE OF,ADVISE,AVAILABILITY,SIDE EFFECT,DRUG INTERACTION,MARKETED WITH OTHER DRUGS,EXAMPLES.


TELMISARTAN



Telmisartan

TELMISARTAN CHEMICAL FORMULA :

C33H30N4O2



TELMISARTAN USES :


used to treat:

high blood pressure (hypertension)





TELMISARTAN MECHANISM OF ACTION :



Telmisartan is an angiotensin II receptor (ARBs) antagonist.



angiotensin II receptor found in

vascular smooth muscle

adrenal gland



angiotensin II receptor role is

vasoconstrictor

stimulates synthesis and release of aldosterone



blockage of angiotensin II receptor results:

relax your veins and arteries to lower your blood pressure

blood can flow more easily



telmisartan is a partial agonist of Peroxisome proliferator-activated receptor gamma (PPARγ).

PPARγ is used as antidiabetic drugs.so telmisartan can improve carbohydrate and lipid metabolism.







TELMISARTAN RECOMMENDED DOSAGE :


(This is ideal dose for your knowledge.Do not take without consult your DOCTOR or PHARMACIST)



As per body weight,condition





TELMISARTAN ADVISE:


SCHEDULE H PRESCRIPTION DRUG-mean- Not to be sold by retail without the prescription of a Registered Medical Practitioner.

Do not take telmisartan if you have ever allergic reaction.

do not stop taking Telmisartan without consulting your doctor even if your blood pressure is controlled. Stopping it suddenly may increase your blood pressure very high.

Telmisartan does not cure high blood pressure but controls it. So, you may have to take the medicine lifetime.

Tell your doctor if you have ever had:

heart problem

kidney disease

liver disease

You should check your potassium levels in blood while you’re taking this drug.



TELMISARTAN AVAILABILITY :


Tablet



TELMISARTAN SIDE EFFECT :


Back Pain

Diarrhea

Body Aches

Muscle Pain

Headache

Dizziness

Nausea



TELMISARTAN DRUG INTERACTION :


Digoxin

Lithium

Aspirin

Angiotensin-converting enzyme (ace) blockers like:


Captopril

Ramipril



Angiotensin receptor ii blockers like:


Losartan



Diuretics like:


Acetazolamide

Chlorothiazide

Ethacrynic acid

Furosemide

Hydrochlorothiazide



Nsaids like:


Diclofenac

Ibuprofen

Naproxen

Piroxicam





TELMISARTAN MARKETED WITH OTHER DRUGS:


Telmisartan + Hydrochlorothiazide

Telmisartan + Metoprolol

Telmisartan + Amlodipine

Telmisartan + Clinidpine

Telmisartan + Chlorthalidone

Telmisartan + Ramipril 























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